I-99% ye-Tianeptine ityuwa yesodium CAS 30123-17-2
Inkcazo
INTO | UMGANGATHO | IZIPHUMO |
Imbonakalo | Umgubo omhlophe ukuya kumthubi | Umgubo omhlophe wekristale |
Ukunyibilika | Inyibilika ngokukhululekileyo Emanzini kunye i-methanol kunye ne-dichloromethane | Iyahambelana |
Ukuchongwa | Nge-IR, Ukuhambelana nomgangatho wokusebenza | Iyahambelana |
(2) Inika ukusabela kwesodium | Iyahambelana | |
Ukungcola A | ≤0.1% | Ayifunyaniswanga |
Iikhompawundi ezinxulumeneyo | Nakuphi na ukungcola okukodwa okuPhezulu≤0.1% | 0.060% |
Ukungcola ngokupheleleyo≤0.4% | 0.36% | |
Intsalela yezinyibilikisi (GC) | I-Acetidin≤ 0.5% | ND |
IDichloromethane≤ 0.06% | ND | |
I-Methanol≤ 0.3% | ND | |
Iacetone≤ 0.5% | 0.29% | |
I-acetonitrile≤0.041% | 0.022% | |
I-Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Amanzi | ≤ 5.0% | 3.8% |
Uvavanyo (HPLC) | 99.0% -101.0% (Kwi-anhydrousbasis) | 99.70% |
Isicelo
I-Tianeptine sodiumityuwai-tricyclic antidepressant.Indlela yayo yokuchasana noxinzelelo yahlukile kuleyo ye-tricyclic antidepressants yesintu.Inokunyusa ukuthathwa kwakhona kwe-5-HT kwi-synaptic cleft.Iziphumo ze-HT neuronal conduction.Akukho budlelwane kwi-choline okanye i-adrenergic receptors.Ukusebenza kwe-antidepressant kufana ne-tricyclics, kodwa ukunyamezela kungcono kunokwe-tricyclics.Kunyango loxinzelelo oluncinci, oluphakathi okanye olunzima, ukudakumba kwe-neurogenic kunye ne-reactive, ukuxhalaba kunye nokudandatheka ngomzimba, ngakumbi ukuphazamiseka kwesisu, kunye nokuxhalaba kunye nokudakumba kwizigulane ezixhomekeke kutywala ngexesha lokuyeka.